SGD Publications 2015 - current

(590).  Asymmetric synthesis of 3-deoxy-3-aminosphingoid bases:approaches based on parallel kinetic resolution
and double asymmetric induction

Csatayová, K.; Davies, S. G.; Fletcher, A. M.; Fowler, T. R.; Kennedy, M. S.; Roberts, P. M.; Thomson, J. E.
J. Org. Chem. 2017, DOI: 10.1021/acs.joc.7b02233 [View Journal Page]

(589).  Stereoselective ammonium-directed epoxidation in the asymmetric syntheses of dihydroconduramines
(−)-A-2, (−)-B-2, (−)-C-3 and (+)-F-3
Da Silva Pinto, S.; Davies, S. G.; Fletcher, A. M.; Roberts, P. M.; Thomson, J. E. Synthesis 2017, in press 

(588).  Asymmetric synthesis of the N-terminal α-hydroxy-β-amino acid components of microginins 612, 646
and 680
Davies, S. G.; Fletcher, A. M.; Hanby, A. R.; Roberts, P. M.; Thomson, J. E. Tetrahedron: Asymmetry 2017,
DOI: 10.1016/j.tetasy.2017.09.022

(587).  Probing competitive and co-operative hydroxyl and ammonium hydrogen-bonding directed epoxidations
Brambilla, M.; Brennan, M. B.; Csatayová, K.; Davies, S. G.; Fletcher, A. M.; Kennett, A. M. R.; Lee, J. A.; Roberts, P. M.; Russell, A. J.; Thomson, J. E. J. Org. Chem. 2017, 82, 10297 [View Journal Page]

(586).  Structural revision of the Hancock alkaloid (−)-galipeine
Davies, S. G.; Fletcher, A. M.; Houlsby, I. T. T.; Roberts, P. M.; Thomson, J. E. J. Org. Chem. 2017, 82, 10673 [View Journal Page]

(585).  Tetrafluoroborate salt fluorination for preparing alkyl fluorides
Davies, S. G.; Roberts P. M. In Synthetic Organofluorine Chemistry. Fluorination; Hu, J.; Umemoto, T., Eds.; Springer, 2017; in press

(584).  Solid state conformations of α,β-unsaturated hydroxamates derived from the ‘chiral Weinreb amide’ auxiliary (S)-N-1-(1'-naphthyl)ethyl-O-tert-butylhydroxylamine
Davies, S. G.; Lee, J. A.; Roberts, P. M.; Thomson, J. E.; Yin, J. Tetrahedron: Asymmetry 2017
DOI: 10.1016/j.tetasy.2017.07.009 [View Journal Page]

(583).  Asymmetric ortho-deprotonation of (η6-arene) chromium tricarbonyl complexes substituted with a chiral hydroxylamine
Da Costa, M. R. G.; Curto, M. J. M.; Davies, S. G.; Teixeira, F. C.; Thomson, J. E. Tetrahedron 2017, 73, 5411 [View Journal Page]

(582).  Regenerative Medicine
Davies, S. G.; Kennewell, P. D.; Russell, A. J.; Silpa, L.; Westwood, R.; Wynne, G. M. In Comprehensive Medicinal Chemistry, III; Chackalamannil, S.; Rotella, D.; Ward, S. Eds.; Elsevier: London, U.K., 2017; 3rd Edn., pp 379–435 [View Abstract]

(581).  Asymmetric synthesis of pyrrolizidines, indolizidines and quinolizidines via a double reductive cyclisation protocol
Davies, S. G.; Fletcher, A. M.; Roberts, P. M.; Thomson, J. E. Synlett 2017, DOI: 10.1055/s-0036-1590975
[View Journal Page]

(580).  Asymmetric synthesis of the tetraponerine alkaloids
Davies, S. G.; Fletcher, A. M.; Houlsby, I. T. T.; Roberts, P. M.; Thomson, J. E. J. Org. Chem. 2017, 82, 6689 [View Journal Page]

(579).  Thiazolidine derivatives as potent and selective inhibitors of the PIM kinase family
Bataille, C. J. R.; Brennan, M. B.; Byrne, S.; Davies, S. G.; Durbin, M.; Fedorov, O.; Huber, K. V. M.; Jones, 
A. M.; Knapp, S.; Liu, G.; Nadali, A.; Quevedo, C. E.; Russell, A. J.; Walker, R. G.; Westwood, R.; Wynne, G. M. Bioorg. Med. Chem. 2017, 25, 2657 [View Journal Page]

(578).  (−)-Pseudodistomin E: first asymmetric synthesis and absolute configuration assignment
Davies, S. G.; Fletcher, A. M.; Roberts, P. M.; Thomson, J. E.; Zimmer, D. Org. Lett. 2017, 19, 1638
[View Journal Page]

(577).  Asymmetric syntheses of the 1-hydroxymethyl-2-hydroxy substituted pyrrolizidines (–)-macronecine,
(–)-petasinecine, (–)-1-epi-macronecine, (+)-1-epi-petasinecine and (+)-2-epi-rosmarinecine
Brambilla, M.; Davies, S. G.; Fletcher, A. M.; Roberts, P. M.; Thomson, J. E. Tetrahedron, 2016, 72, 7449
[View Journal Page]

(576).  Pyrrolizidines, indolizidines and quinolizidines via a double reductive cyclisation protocol: concise asymmetric syntheses of (+)-trachelanthamidine, (+)-tashiromine and (+)-epilupinine
Brambilla, M.; Davies, S. G.; Fletcher, A. M.; Roberts, P. M.; Thomson, J. E.; Zimmer, D. Tetrahedron 2016,
72, 7417 [View Journal Page]

(575).  Asymmetric syntheses of (–)-ADMJ and (+)-ADANJ: 2-deoxy-2-amino analogues of
(–)-1-deoxymannojirimycin and (+)-1-deoxyallonojirimycin
Davies, S. G.; Figuccia A. L. A.; Fletcher, A. M.; Roberts, P. M.; Thomson, J. E. J. Org. Chem. 2016, 81, 6481 [View Journal Page]

(574).  Asymmetric syntheses of (–)-hastanecine, (–)-turneforcidine and (–)-platynecine
Brambilla, M.; Davies, S. G.; Fletcher, A. M.; Roberts, P. M.; Thomson, J. E. Tetrahedron 2016, 72, 4523
[View Journal Page]

(573).  Asymmetric syntheses of (+)-preussin B, the C(2)-epimer of (–)-preussin B, and 3-deoxy-(+)-preussin B
Buchman, M.; Csatayová, K.; Davies, S. G.; Fletcher, A. M.; Houlsby, I. T. T.; Roberts, P. M.; Rowe, S.; Thomson, J. E. J. Org. Chem. 2016, 81, 4907 [View Journal Page]

(572).  Strategies for the construction of morphinan alkaloid AB-rings: regioselective Friedel-Crafts-type cyclisations of γ-aryl-β-benzoylamido acids with asymmetrically substituted γ-aryl rings
Davies, S. G.; Goddard, E, C.; Roberts, P. M.; Russell, A. J.; Smith, A. D.; Thomson, J. E.; Withey, J. M. Tetrahedron: Asymmetry 2016, 27, 274 [View Journal Page]

(571).  Trading N and O. Part 3: Synthesis of 1,2,3,4-tetrahydroisoquinolines from α-hydroxy-β-amino esters
Davies, S. G.; Fletcher, A. M.; Frost, A. B.; Kennedy, M. S.; Roberts, P. M.; Thomson, J. E. Tetrahedron 2016, 72, 2139 [View Journal Page]

(570).  Asymmetric synthesis of N,O-diacetyl-3-epi-xestoaminol C: structure and absolute configuration confirmation of 3-epi-xestoaminol C
Archer, S. G.; Csatayová, K.; Davies, S. G.; Fletcher, A. M.; Roberts, P. M.; Thomson, J. E. Tetrahedron Lett. 2016, 57, 1270 [View Journal Page]

(569).  The asymmetric synthesis of enantiopure C(5)-substituted transpentacins via diastereoselective conjugate additions to a β'-amino-α,β-unsaturated ester
Davies, S. G.; Fletcher, A. M.; Roberts, P. M.; Thomson, J. E.; Zammit, C. M. Tetrahedron: Asymmetry 2016,
27, 208 [View Journal Page]

(568).  Asymmetric syntheses of the methyl 3-deoxy-3-amino-glycosides of D-glycero-L-gulo-heptose, D-glycero-D-galacto-heptose, D-glycero-L-allo-heptose and D-glycero-D-allo-heptose
Brambilla, M.; Davies, S. G.; Diment, W. T.; Fletcher, A. M.; Lee, J. A.; Roberts, P. M.; Thomson, J. E.; Waul,
M. A. Tetrahedron: Asymmetry 2016, 27, 31 [View Journal Page]

(567).  Syntheses of (R)-sitagliptin
Davies, S. G.; Fletcher, A. M.; Thomson, J. E. Tetrahedron: Asymmetry 201526, 1109 [View Journal Page]

(566).  Asymmetric syntheses of polysubstituted homoprolines and homoprolinols
Csatayová, K.; Davies, S. G.; Figuccia, A. L. A.; Fletcher, A. M.; Ford, J. G.; Lee, J. A.; Roberts, P. M.;
Saward, B. G.; Song, H.; Thomson, J. E. 
Tetrahedron 201571, 9131 [View Journal Page]

(565).  Synthesis and crystal structures of 2-azido-4-aminocyclohexane-1,3-diols
Brennan, M. B.; Davies, S. G.; Lee, J. A.; Thompson, A. L.; Thomson, J. E. J. Chem. Crystallogr. 2015,
45, 401 [View Journal Page]

(564).  Second-generation compound for the modulation of utrophin in the therapy of DMD
Guiraud, S.; Squire, S. E.; Edwards, B.; Chen, H.; Burns, D. T.; Shah, N.; Babbs, A.; Davies, S. G.; Wynne, G. M.; Russell, A. J.; Elsey, D.; Wilson, F. X.; Tinsley, J. M.; Davies, K. E. Hum. Mol. Genet. 201524, 4212
[View Journal Page]

(563).  Syntheses of dihydroconduramines (±)-B-1, (±)-E-1 and (±)-F-1 via diastereoselective epoxidation of
N-protected 4-aminocyclohex-2-en-1-ols
Brennan, M.; Csatayov
á, K.; Davies, S. G.; Fletcher, A. M.; Green, W. D.; Lee, J. A.; Roberts, P. M.; Russell, A. J.; Thomson, J. E. J. Org. Chem. 201580, 6609 [View Journal Page]

(562).  Enantiopure 3-amino substituted 1-indanones, 1-tetralones and 1-benzosuberones via Friedel-Crafts cyclisation of ω-aryl-β-benzamido acids
Davies, S. G.; Goddard, E. C.; Roberts, P. M.; Russell, A. J.; Thomson, J. E Synlett 201526, 1541
[View Journal Page]

(561).  Asymmetric synthesis of substituted anti-β-fluorophenylalanines
Davies, S. G.; Fletcher, A. M.; Frost, A. B.; Roberts, P. M.; Thomson, J. E. Org. Lett. 201517, 2254
[View Journal Page]

(560).  Asymmetric syntheses of nakinadine D, nakinadine E and nakinadine F: confirmation of their relative (RS,SR)-configurations and proposal of their absolute (2S,3R)-configurations
Davies, S. G.; Fletcher, A. M.; Shah, R. S.; Roberts, P. M.; Thomson, J. E. J. Org. Chem. 201580, 4017
[View Journal Page]

(559).  Conformational analysis of triphenylphosphine ligands in stereogenic monometallic complexes: tools for predicting the preferred configuration of the triphenylphosphine rotor
Costello, J. F.; Davies, S. G.; Gould, E. T. F.; Thomson, J. E. Dalton Trans. 201544, 5451 [View Journal Page]

(558).  Diastereoselective conjugate additions to alkoxycarbene cations of the iron chiral auxiliary
[(η5-C5H5)Fe(CO)(PPh3)=C(OMe)CH=CHR]+
Davies, S. G.; Easton, R. J. C.; McKenna, J. M; Polywka, M. E. C; Thomson, J. E. J. Organomet. Chem. 2015,
792, 66 [View Journal Page]

(557).  Stemistry: the control of stem cells in situ using chemistry
Davies, S. G.; Kennewell, 
P. D.; Russell, A. J.; Seden, P. T.; Westwood, R.; Wynne, G. M. J. Med. Chem. 201558, 2863 [View Journal Page]

(556).  Pinacolatoboron fluoride (pinBF) is an efficient fluoride transfer agent for synthesis of benzylic fluorides
Cresswell, A. J.; Davies, S. G.; Figuccia, A. L. A.; Fletcher, A. M.; Heijnen, D.; Lee, J. A.; Morris, M. J.; Kennett,
A. M. R.; Roberts, P. M.; Thomson, J. E. Tetrahedron Lett. 201556, 3373 [View Journal Page]

(555).  Concise total asymmetric syntheses of (–)-fagomine, two of its epimers, and two seven-membered
ring congeners
Csatayová, K.; Davies, S. G.; Fletcher, A. M.; Ford, J. G.; Klauber, D. J.; Roberts, P. M. Thomson, J. E. Tetrahedron 201571, 7170 [View Journal Page]

(554).  Epoxidation of trans-4-aminocyclohex-2-en-1-ol derivatives: competition of hydroxyl-directed and ammonium-directed pathways
Brennan, M. B.; Davies, S. G.; Fletcher, A. M.; Lee, J. A.; Roberts, P. M.; Russell, A. J.; Thomson, J. E.
Aust. J. Chem. 201568, 610 [View Journal Page]

(553).  Beyond the Balz-Schiemann reaction: the utility of tetrafluoroborates and boron trifluoride as nucleophilic fluoride sources
Davies, S. G.; Roberts, P. M.; Cresswell, A. J.; Thomson, J. E. Chem. Rev. 2015115, 566 [View Journal Page]

(552).  The homalium alkaloids: isolation, synthesis and absolute configuration assignment
Davies, S. G.; Thomson J. E. In The Alkaloids: Chemistry and Biology; Knölker, H.-J., Ed.; Elsevier: London, U.K., 2015; Vol. 74, pp 121–158 [View Abstract]

 

 

 

 


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